A Fast and Efficient Method for the Synthesis of 1,5-Benzodiazepine Derivatives Under Solvent-Free Conditions

نویسندگان

  • Ahmad Shaabani Department of Chemistry, Shahid Beheshti University, P.O. Box 19396-4717 Tehran, I.R. IRAN
  • Ali Maleki Department of Chemistry, Shahid Beheshti University, P.O. Box 19396-4717 Tehran, I.R. IRAN
چکیده مقاله:

Silica sulfuric acid is found to catalyze efficiently the condensation of o-phenylenediamines with various linear and cyclic ketones to afford the corresponding 1,5-benzodiazepines in quantitative yields under solvent-free conditions at room temperature

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a fast and efficient method for the synthesis of 1,5-benzodiazepine derivatives under solvent-free conditions

silica sulfuric acid is found to catalyze efficiently the condensation of o-phenylenediamines with various linear and cyclic ketones to afford the corresponding 1,5-benzodiazepines in quantitative yields under solvent-free conditions at room temperature

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عنوان ژورنال

دوره 26  شماره 4

صفحات  93- 97

تاریخ انتشار 2007-12-01

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